Sodium Caffeine Benzoate


Composition 1 Sodium Caffeine Benzoate may include 100 mg or 200 mg caffeine. Additional substances: calcium stearate, potato starch.

In 1 ml Caffeine Benzoate Sodium contains 200 mg caffeine. Additional substances: water, sodium chloride.

Release form

  • 6 or 10 tablets per cell;
  • 6 or 10 tablets in a non-cell package;
  • 1 ml solution in ampoules; 10 ampoules in a pack of cardboard.

Pharmachologic effect

Psychostimulant, cardiotonic, analeptic act.

Pharmacodynamics and pharmacokinetics

Pharmacopoeia relates this medicine to analeptic and psychostimulating. Derived methylxanthine.Inhibits peripheral and central receptors adenosinein a competitive way. Inhibits activity phosphodiesterase in the heart, nervous system, skeletal muscles, adipose tissue, smooth muscle organs, enhances the accumulation in them cGMP and cAMP (when used only in large doses). Activates the respiratory and vasomotor centers of the midbrain, as well as the core n.vagushas a direct stimulating effect on the cortex. In high doses, it improves interneuronal conduction, enhancing reflexes at the level of the spinal cord.

Stimulates physical and mental performance, activates mental activity, motor activity, reduces reaction time, reduces fatigue and drowsiness for a while. When taken in small doses, the effect of neurostimulation predominates, and in large doses, suppression of the nervous system.

Makes breathing deeper and increases its frequency. It usually has a positive chrono-, batmo-, foreign- and dromotropic effect. It stimulates the vasomotor core and has a relaxing effect on the vessel wall, which causes the expansion of arteries and veins of the kidneys, skeletal muscles, heart, and the tone of the arteries of the brain increases.

Pressure changes under the influence of cardiac and vascular mechanisms of action caffeine: at normal pressure caffeine does not change or slightly increases it, with initially reduced - normalizes it.

It has a relaxing effect on smooth muscles (including bronchi), and on skeletal - stimulating. Enhances secretory function of the stomach. It has a diuretic effect, which is due to a decrease in the reverse absorption of sodium ions and water molecules in the renal tubules, as well as a relaxation of the walls of the vessels of the kidneys and increased filtration in the glomeruli of the kidneys. Weakens aggregation platelet count and exit histaminefrom macrophages. Stimulates processes glycogenolysisand lipolysis.

Indications for use

  • decreased performance (physical and mental);
  • disorders that occur with inhibition of nervous activity, the work of the cardiovascular and respiratory systems (including overdose opioid analgesics and diseases of an infectious nature);
  • cerebrovascular spasms;
  • drowsiness.


  • organic lesions of the circulatory system (including severe atherosclerosis);
  • arterial hypertension;
  • increased irritability;
  • senile age;
  • glaucoma;
  • sleep disturbances.

Side effects

  • Disorders from nervous system: anxiety, agitation, sleep disturbance, with prolonged use addiction is not excluded.
  • Disorders from blood circulation: pressure increase, arrhythmias, tachycardia.
  • Disorders from digestion: vomiting, nausea.

Sodium Caffeine Benzoate Instruction (Method and Dosage)

The solution in ampoules is administered subcutaneously, and the sodium caffeine-benzoate tablets are taken orally. Adults are prescribed 100-200 mg of the drug up to three times a day, and for children - 25-100 mg also up to three times a day.


Signs of an overdose: agitation, anxiety, motor anxiety, agitation, muscle twitching, tremor, hyperesthesia, epileptic seizures, ciliary scotoma, headacheringing in the ears, confusion, insomnia, rave, tachycardia, delirium, arrhythmia, frequent urination hyperthermia dehydration, vomiting, nausea.

Overdose treatment: breath support, oxygenation, hemodialysis, regulation of fluid and electrolyte balance, prescribed for epileptic seizures Diazepam, Phenytoinor Phenobarbital intravenously.


When used together, the effects of sleeping pills and drugs for anesthesia are reduced.

When combined, amplification of effects is possible analgesics, antipyretics, Naproxen, Salicylamide.

While using estrogen amplification and increase in duration of action is possible caffeine due to inhibition isoenzyme CYP1A2.

When combined with adenosine it is possible that a decrease in the increased number of heart contractions caused by the introduction of Adenosine; the drug also reduces vasodilation associated with the action Adenosine.

When combined with acetylsalicylic acid it is possible to increase its absorption rate, bioavailability and concentration in blood.

While using Mexiletine reduces clearance caffeine and increases its plasma content by blocking metabolism last in the liver.

Methoxalen slows down caffeine with the possible stimulation of its effect and the appearance of toxic effects.

Due to the activation of microsomal enzymes under the influence of Phenytoin when it is taken together, the exchange and excretion are accelerated caffeine.

Terbinafine, Ketoconazole and Fluconazole moderately increase concentration caffeine in blood.

While taking caffeineaccelerates absorption ergotamine.

Terms of sale

Without recipe.

Storage conditions

Keep out of the reach of children. Store at temperatures up to 25 ° C.

Shelf life

5 years.

Special instructions

The effect on the central nervous system can be expressed by excitation or, conversely, inhibition, depending on its type.

Use with caution in patients with peptic ulcer.

For children

The drug is not used in children under 12 years of age.

For weight loss

Caffeine often used for weight loss. This is due to a decrease appetite and increased physical stamina when using the drug. Some nutritionists indicate ability caffeine burn an additional 5 kg of weight per month amid intense physical training. It is worth remembering that the uncontrolled use of the drug can cause unwanted side effects.

During pregnancy and lactation

The drug is not used in these periods.

Sodium Caffeine Benzoate Reviews

Reviews characterize the drug as an effective means to maintain and improve performance when used in moderation. You should always remember that uncontrolled administration of the drug can lead to the development of an overdose and serious side effects.

Price Sodium Caffeine Benzoate, where to buy

The price of 100 mg tablets No. 6 can reach 40 rubles in Russia. You can buy 200 mg No. 10 in Ukraine for 15 hryvnias.

  • Online Pharmacies in Russia
  • Online pharmacies in UkraineUkraine
  • Online pharmacies in Kazakhstan


  • Sodium caffeine benzoate tab. 100mg n10AO Tatkhimpharmpreparaty56 rub.order
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  • Sodium caffeine-benzoate 0.2 №10 tablets TOV "Agrofarm", Ukraine19 UAH order
  • Sodium caffeine-benzoate 10% 1 ml No. 10 solution for injection TOV "Dosledniy Zavod GNTsLS", Ukraine / TOV "FC" Zdorovya ", Ukraine19 UAH order
  • Caffeine-sodium benzoate 10% 1 ml №10 injection for 21 UAH order

Pani Pharmacy

  • Sodium caffeine-benzoate ampoule Caffeine-benzoate sodium solution d / in. 10% 1ml №10 Ukraine, Darnitsa PrJSC 22 UAH order
  • Sodium caffeine-benzoate ampoule Caffeine-benzoate sodium solution d / in. 10% 1ml №10 Ukraine, OZ GNTsLS LLC 18 UAH order
  • Sodium caffeine-benzoate ampoule Caffeine-benzoate sodium solution d / in. 20% 1ml №10 Ukraine, OZ GNTsLS LLC 27 UAH to order
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  • Caffeine-benzoate sodium 20% / 1 ml No. 10 solution for in. amp. Borisov ZMP (Belarus) 240 tg.order
  • Caffeine-sodium benzoate-Darnitsa 10% / 1 ml No. 10 solution for in. amp. Darnitsa (Ukraine) 195 tg.order
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